A single M1 residue in the beta2 subunit alters channel gating of GABAA receptor in anesthetic modulation and direct activation. [electronic resource]
- The Journal of biological chemistry Oct 2003
- 42821-8 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
0021-9258
10.1074/jbc.M306978200 doi
Adjuvants, Anesthesia--pharmacology Allosteric Site Amino Acid Sequence Anesthetics--pharmacology Anesthetics, Intravenous--pharmacology Animals Cloning, Molecular DNA Mutational Analysis Dose-Response Relationship, Drug Etomidate--pharmacology Kinetics Ligands Models, Biological Molecular Sequence Data Mutagenesis Mutation Oocytes--metabolism Patch-Clamp Techniques Pentobarbital--pharmacology Point Mutation Pregnanediones--pharmacology Propofol--pharmacology Protein Structure, Tertiary RNA, Messenger--metabolism Rats Receptors, GABA-A--chemistry Recombinant Proteins--metabolism Xenopus