Campiani, Giuseppe

Synthesis and pharmacological evaluation of potent and highly selective D3 receptor ligands: inhibition of cocaine-seeking behavior and the role of dopamine D3/D2 receptors. [electronic resource] - Journal of medicinal chemistry Aug 2003 - 3822-39 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-2623

10.1021/jm0211220 doi


Animals
Behavior, Addictive--drug therapy
Brain--metabolism
Cocaine--administration & dosage
Cocaine-Related Disorders--psychology
Conditioning, Operant--drug effects
Dopamine Agonists--chemical synthesis
Dopamine Antagonists--chemical synthesis
Extinction, Psychological--drug effects
In Vitro Techniques
Ligands
Male
Models, Molecular
Piperazines--chemical synthesis
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptors, Dopamine D2--drug effects
Receptors, Dopamine D3
Self Administration
Structure-Activity Relationship