Non-nucleoside inhibitors of HIV-1 reverse transcriptase inhibit phosphorolysis and resensitize the 3'-azido-3'-deoxythymidine (AZT)-resistant polymerase to AZT-5'-triphosphate. [electronic resource]
- The Journal of biological chemistry Oct 2003
- 42710-6 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0021-9258
10.1074/jbc.M212673200 doi
Adenosine Triphosphate--pharmacology Anti-HIV Agents--pharmacology Dideoxynucleotides Diphosphates--pharmacology Drug Resistance, Viral Drug Synergism Drug Therapy, Combination HIV Reverse Transcriptase--drug effects Humans Mutation, Missense Nevirapine--pharmacology Phosphorylation--drug effects Protein Subunits--genetics Reverse Transcriptase Inhibitors--pharmacology Thymine Nucleotides--pharmacology Zidovudine--analogs & derivatives