Amos, Gregory J

Block of HERG-carried K+ currents by the new repolarization delaying agent H 345/52. [electronic resource] - Journal of cardiovascular electrophysiology Jun 2003 - 651-8 p. digital

Publication Type: Comparative Study; Evaluation Study; Journal Article

1045-3873

10.1046/j.1540-8167.2003.02554.x doi


Action Potentials--drug effects
Alkanes--administration & dosage
Animals
Anti-Arrhythmia Agents--pharmacology
Binding, Competitive--drug effects
Bridged Bicyclo Compounds--administration & dosage
Cation Transport Proteins
Cell Line
DNA-Binding Proteins
Dose-Response Relationship, Drug
ERG1 Potassium Channel
Ether-A-Go-Go Potassium Channels
Fibroblasts--drug effects
Heart--physiology
Humans
Inhibitory Concentration 50
Membrane Potentials--drug effects
Mice
Models, Animal
Patch-Clamp Techniques
Phenethylamines--pharmacology
Potassium Channel Blockers--pharmacology
Potassium Channels--drug effects
Potassium Channels, Voltage-Gated
Predictive Value of Tests
Propanolamines--pharmacology
Sulfonamides--pharmacology
Time Factors
Trans-Activators
Transcriptional Regulator ERG