Anti-androgens with full antagonistic activity toward human prostate tumor LNCaP cells with mutated androgen receptor. [electronic resource]
- Bioorganic & medicinal chemistry letters Aug 2003
- 2655-8 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0960-894X
10.1016/s0960-894x(03)00575-4 doi
Androgen Antagonists--chemical synthesis Binding, Competitive Drug Design Humans Isoxazoles--chemical synthesis Male Molecular Structure Point Mutation Prostate-Specific Antigen--analysis Protein Folding Receptors, Androgen--biosynthesis Testosterone Tumor Cells, Cultured