Ishioka, Toshiyasu

Anti-androgens with full antagonistic activity toward human prostate tumor LNCaP cells with mutated androgen receptor. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2003 - 2655-8 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

0960-894X

10.1016/s0960-894x(03)00575-4 doi


Androgen Antagonists--chemical synthesis
Binding, Competitive
Drug Design
Humans
Isoxazoles--chemical synthesis
Male
Molecular Structure
Point Mutation
Prostate-Specific Antigen--analysis
Protein Folding
Receptors, Androgen--biosynthesis
Testosterone
Tumor Cells, Cultured