Design and synthesis of poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors. Part 3: In vitro evaluation of 1,3,4,5-tetrahydro-benzo[c][1,6]- and [c][1,7]-naphthyridin-6-ones. [electronic resource]
- Bioorganic & medicinal chemistry letters Aug 2003
- 2513-8 p. digital
Publication Type: Journal Article
0960-894X
10.1016/s0960-894x(03)00465-7 doi
Chemical Phenomena Chemistry, Physical Enzyme Inhibitors--chemical synthesis Indicators and Reagents Naphthyridines--chemical synthesis Poly(ADP-ribose) Polymerase Inhibitors Solubility Structure-Activity Relationship