The human multidrug resistance protein MRP4 functions as a prostaglandin efflux transporter and is inhibited by nonsteroidal antiinflammatory drugs. [electronic resource]
- Proceedings of the National Academy of Sciences of the United States of America Aug 2003
- 9244-9 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0027-8424
10.1073/pnas.1033060100 doi
Adenosine Triphosphate--metabolism Alprostadil--metabolism Animals Anti-Inflammatory Agents, Non-Steroidal--pharmacology Biological Transport Cell Line Cell Membrane--metabolism Diffusion Dinoprost--metabolism Dinoprostone--metabolism Dose-Response Relationship, Drug Humans Insecta Multidrug Resistance-Associated Proteins Prostaglandins--metabolism Prostaglandins A--metabolism Prostaglandins F--metabolism RNA Interference RNA, Small Interfering--metabolism Ribosomal Proteins--chemistry Thromboxane B2--metabolism Time Factors