TY - GEN AU - MacKenzie,A Roderick AU - Marchington,Allan P AU - Middleton,Donald S AU - Newman,Sandra D AU - Selway,Christopher N AU - Terrett,Nicholas K TI - 4-Amino-2-(aryl)-butylbenzamides and Their conformationally constrained analogues. Potent antagonists of the human neurokinin-2 (NK(2)) receptor SN - 0960-894X PY - 2004///0301 KW - Animals KW - Benzamides KW - chemical synthesis KW - CHO Cells KW - Cricetinae KW - Cyclization KW - Drug Design KW - Duodenum KW - drug effects KW - Humans KW - In Vitro Techniques KW - Molecular Conformation KW - Peptide Library KW - Piperidines KW - Rats KW - Receptors, Neurokinin-2 KW - antagonists & inhibitors KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/s0960-894x(03)00343-3 ER -