Relationships between the hydrophilic-lipophilic balance values of pharmaceutical excipients and their multidrug resistance modulating effect in Caco-2 cells and rat intestines. [electronic resource]
- Journal of controlled release : official journal of the Controlled Release Society Jun 2003
- 37-48 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0168-3659
10.1016/s0168-3659(03)00163-9 doi
Adjuvants, Pharmaceutic--chemistry Animals Antibiotics, Antineoplastic--pharmacokinetics Biological Transport--drug effects Caco-2 Cells Drug Resistance, Multiple Drug Resistance, Neoplasm Electric Conductivity Epirubicin--pharmacokinetics Excipients--chemistry Humans Ileum--drug effects In Vitro Techniques Intestinal Absorption--drug effects Intestinal Mucosa--metabolism Intestines--drug effects Jejunum--drug effects Male Rats Rats, Sprague-Dawley