Schlechtingen, Georg

Structure-activity relationships of dynorphin a analogues modified in the address sequence. [electronic resource] - Journal of medicinal chemistry May 2003 - 2104-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0022-2623

10.1021/jm020125+ doi


Analgesics, Opioid--chemical synthesis
Animals
CHO Cells
Cricetinae
Dynorphins--chemistry
Guanosine 5'-O-(3-Thiotriphosphate)--pharmacology
Guinea Pigs
Ileum--drug effects
In Vitro Techniques
Muscle Contraction--drug effects
Muscle, Smooth--drug effects
Oligopeptides--chemical synthesis
Radioligand Assay
Receptors, Opioid, delta--metabolism
Receptors, Opioid, kappa--agonists
Receptors, Opioid, mu--metabolism
Structure-Activity Relationship