Zhu, Guoxin

Synthesis, structure-activity relationship, and biological studies of indolocarbazoles as potent cyclin D1-CDK4 inhibitors. [electronic resource] - Journal of medicinal chemistry May 2003 - 2027-30 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm0256169 doi


Antineoplastic Agents--chemical synthesis
Carbazoles--chemical synthesis
Cell Division--drug effects
Cyclin D1--metabolism
Cyclin-Dependent Kinase 4
Cyclin-Dependent Kinases--antagonists & inhibitors
Drug Screening Assays, Antitumor
Enzyme Inhibitors--chemical synthesis
G1 Phase--drug effects
Humans
Indoles--chemical synthesis
Phosphorylation
Proto-Oncogene Proteins
Retinoblastoma Protein--metabolism
Structure-Activity Relationship
Tumor Cells, Cultured