Expression of the human CYP3A4 gene in the small intestine of transgenic mice: in vitro metabolism and pharmacokinetics of midazolam. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals May 2003
- 548-58 p. digital
Publication Type: Journal Article
0090-9556
10.1124/dmd.31.5.548 doi
Administration, Oral Animals Area Under Curve Biological Availability Blotting, Southern Cytochrome P-450 CYP3A Cytochrome P-450 Enzyme System--genetics Dexamethasone--pharmacology Drug Interactions Enzyme Inhibitors--pharmacology Half-Life Humans In Vitro Techniques Intestine, Small--metabolism Ketoconazole--pharmacology Male Mice Mice, Transgenic Microsomes--drug effects Midazolam--analogs & derivatives Polymerase Chain Reaction Rifampin--pharmacology Time Factors