SSR591813, a novel selective and partial alpha4beta2 nicotinic receptor agonist with potential as an aid to smoking cessation. [electronic resource]
- The Journal of pharmacology and experimental therapeutics Jul 2003
- 407-20 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-3565
10.1124/jpet.103.049262 doi
Animals Azepines--therapeutic use Behavior, Animal--drug effects Body Temperature--drug effects Brain--metabolism Cardiovascular System--drug effects Cells, Cultured Dextroamphetamine--pharmacology Discrimination Learning Drug Interactions Heterocyclic Compounds, 4 or More Rings--therapeutic use Humans Male Mecamylamine--pharmacology Microdialysis Motor Activity--drug effects Nicotine--pharmacology Nicotinic Agonists--therapeutic use Oocytes--drug effects Radioligand Assay Rats Rats, Sprague-Dawley Receptors, Nicotinic--drug effects Self Administration Smoking--drug therapy Smoking Cessation Substance Withdrawal Syndrome Transfection Xenopus laevis