Cohen, C

SSR591813, a novel selective and partial alpha4beta2 nicotinic receptor agonist with potential as an aid to smoking cessation. [electronic resource] - The Journal of pharmacology and experimental therapeutics Jul 2003 - 407-20 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-3565

10.1124/jpet.103.049262 doi


Animals
Azepines--therapeutic use
Behavior, Animal--drug effects
Body Temperature--drug effects
Brain--metabolism
Cardiovascular System--drug effects
Cells, Cultured
Dextroamphetamine--pharmacology
Discrimination Learning
Drug Interactions
Heterocyclic Compounds, 4 or More Rings--therapeutic use
Humans
Male
Mecamylamine--pharmacology
Microdialysis
Motor Activity--drug effects
Nicotine--pharmacology
Nicotinic Agonists--therapeutic use
Oocytes--drug effects
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptors, Nicotinic--drug effects
Self Administration
Smoking--drug therapy
Smoking Cessation
Substance Withdrawal Syndrome
Transfection
Xenopus laevis