Engineering exosite peptides for complete inhibition of factor VIIa using a protease switch with substrate phage. [electronic resource]
- The Journal of biological chemistry Jun 2003
- 21823-30 p. digital
Publication Type: Journal Article
0021-9258
10.1074/jbc.M300951200 doi
Amino Acid Sequence Amino Acids--chemistry Anticoagulants--pharmacology Arginine--chemistry Binding Sites Crystallography, X-Ray DNA--metabolism Dose-Response Relationship, Drug Factor VIIa--antagonists & inhibitors Humans Hydrogen-Ion Concentration Inhibitory Concentration 50 Models, Biological Models, Molecular Molecular Sequence Data Peptide Library Peptides--chemistry Protein Binding Protein Structure, Tertiary Prothrombin Time Thromboplastin--chemistry