Zhang, Puwen
Novel 6-aryl-1,4-dihydrobenzo[d]oxazine-2-thiones as potent, selective, and orally active nonsteroidal progesterone receptor agonists. [electronic resource]
- Bioorganic & medicinal chemistry letters Apr 2003
- 1313-6 p. digital
Publication Type: Journal Article
0960-894X
10.1016/s0960-894x(03)00128-8 doi
Alkaline Phosphatase--biosynthesis
Animals
Breast Neoplasms--enzymology
Cross Reactions
Decidua--drug effects
Female
Humans
Medroxyprogesterone Acetate--pharmacology
Ovariectomy
Oxazines--chemical synthesis
Rats
Receptors, Androgen--drug effects
Receptors, Glucocorticoid--drug effects
Receptors, Progesterone--agonists
Structure-Activity Relationship
Thiones--chemical synthesis