TY - GEN AU - Baraldi,Pier Giovanni AU - Fruttarolo,Francesca AU - Tabrizi,Mojgan Aghazadeh AU - Preti,Delia AU - Romagnoli,Romeo AU - El-Kashef,Hussein AU - Moorman,Allan AU - Varani,Katia AU - Gessi,Stefania AU - Merighi,Stefania AU - Borea,Pier Andrea TI - Design, synthesis, and biological evaluation of C9- and C2-substituted pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as new A2A and A3 adenosine receptors antagonists SN - 0022-2623 PY - 2003///0502 KW - Animals KW - Binding, Competitive KW - Cricetinae KW - Drug Design KW - Humans KW - Molecular Conformation KW - Purinergic P1 Receptor Antagonists KW - Pyrazoles KW - chemical synthesis KW - Pyrimidines KW - Radioligand Assay KW - Receptor, Adenosine A2A KW - Receptor, Adenosine A3 KW - Solubility KW - Structure-Activity Relationship N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1021/jm021023m ER -