Parkes, Kevin E B

Use of a pharmacophore model to discover a new class of influenza endonuclease inhibitors. [electronic resource] - Journal of medicinal chemistry Mar 2003 - 1153-64 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm020334u doi


Animals
Antiviral Agents--chemical synthesis
Binding Sites
Butyrates--chemical synthesis
Cell Line
Combinatorial Chemistry Techniques
DNA-Directed RNA Polymerases--chemistry
Databases, Factual
Dogs
Endonucleases--antagonists & inhibitors
Enzyme Inhibitors--chemical synthesis
Heterocyclic Compounds, 3-Ring--chemical synthesis
Heterocyclic Compounds, 4 or More Rings--chemical synthesis
Influenza A virus--drug effects
Influenza B virus--drug effects
Keto Acids--chemical synthesis
Models, Molecular
Phthalimides--chemical synthesis
Protein Binding
Structure-Activity Relationship