[3H]-methoxymethyl-MTEP and [3H]-methoxy-PEPy: potent and selective radioligands for the metabotropic glutamate subtype 5 (mGlu5) receptor. [electronic resource]
- Bioorganic & medicinal chemistry letters Feb 2003
- 351-4 p. digital
Publication Type: Journal Article
0960-894X
10.1016/s0960-894x(02)00997-6 doi
Animals Binding Sites Brain--drug effects Chemical Phenomena Chemistry, Physical Humans In Vitro Techniques Ligands Male Pyridines--pharmacokinetics Radiopharmaceuticals--pharmacokinetics Rats Receptor, Metabotropic Glutamate 5 Receptors, Metabotropic Glutamate--drug effects Thiazoles--pharmacokinetics