Ding, Zhongren

Inactivation of the human P2Y12 receptor by thiol reagents requires interaction with both extracellular cysteine residues, Cys17 and Cys270. [electronic resource] - Blood May 2003 - 3908-14 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

0006-4971

10.1182/blood-2002-10-3027 doi


4-Chloromercuribenzenesulfonate--pharmacology
Adenosine Diphosphate--pharmacology
Amino Acid Sequence
Animals
Base Sequence
Binding Sites
CHO Cells
Cricetinae
Cyclic AMP--metabolism
Cysteine
DNA Primers
Humans
Inositol Phosphates--metabolism
Kinetics
Membrane Proteins
Molecular Sequence Data
Purinergic P2 Receptor Antagonists
Receptors, Purinergic P2--chemistry
Receptors, Purinergic P2Y1
Receptors, Purinergic P2Y12
Recombinant Proteins--antagonists & inhibitors
Sequence Alignment
Sequence Homology, Amino Acid
Sulfhydryl Compounds--pharmacology
Transfection