Feling, Robert H

Salinosporamide A: a highly cytotoxic proteasome inhibitor from a novel microbial source, a marine bacterium of the new genus salinospora. [electronic resource] - Angewandte Chemie (International ed. in English) Jan 2003 - 355-7 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

1433-7851

10.1002/anie.200390115 doi


Actinomycetales--chemistry
Adenocarcinoma--metabolism
Colonic Neoplasms--metabolism
Crystallography, X-Ray
Cysteine Endopeptidases
Humans
Inhibitory Concentration 50
Lactones--chemistry
Magnetic Resonance Spectroscopy
Models, Molecular
Molecular Structure
Multienzyme Complexes--antagonists & inhibitors
Protease Inhibitors--chemistry
Proteasome Endopeptidase Complex
Pyrroles
Tumor Cells, Cultured