TY  - GEN
AU  - MacKenzie,A Roderick
AU  - Marchington,Allan P
AU  - Middleton,Donald S
AU  - Newman,Sandra D
AU  - Jones,Barry C
TI  - Structure-activity relationships of 1-alkyl-5-(3,4-dichlorophenyl)- 5-[2-[(3-substituted)-1-azetidinyl]ethyl]-2-piperidones. 1. Selective antagonists of the neurokinin-2 receptor
SN  - 0022-2623
PY  - 2002///1220
KW  - Animals
KW  - Azetidines
KW  - chemical synthesis
KW  - CHO Cells
KW  - Cricetinae
KW  - Drug Stability
KW  - Humans
KW  - In Vitro Techniques
KW  - Microsomes, Liver
KW  - metabolism
KW  - Muscle Contraction
KW  - drug effects
KW  - Muscle, Smooth
KW  - Piperazines
KW  - Piperidones
KW  - Pulmonary Artery
KW  - Rabbits
KW  - Radioligand Assay
KW  - Receptors, Neurokinin-2
KW  - antagonists & inhibitors
KW  - Receptors, Neurokinin-3
KW  - Stereoisomerism
KW  - Structure-Activity Relationship
N1  - Publication Type: Journal Article
UR  - https://doi.org/10.1021/jm0209331
ER  -