The molecular and enzyme kinetic basis for the diminished activity of the cytochrome P450 2D6.17 (CYP2D6.17) variant. Potential implications for CYP2D6 phenotyping studies and the clinical use of CYP2D6 substrate drugs in some African populations. [electronic resource]
- Biochemical pharmacology Nov 2002
- 1387-98 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0006-2952
10.1016/s0006-2952(02)01351-5 doi
Africa Alleles Amino Acid Sequence Binding, Competitive Cytochrome P-450 CYP2D6--genetics Genetics, Population Humans Kinetics Models, Biological Models, Molecular Molecular Sequence Data Phenotype Sequence Homology, Amino Acid