Wissner, Allan

Syntheses and EGFR and HER-2 kinase inhibitory activities of 4-anilinoquinoline-3-carbonitriles: analogues of three important 4-anilinoquinazolines currently undergoing clinical evaluation as therapeutic antitumor agents. [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2002 - 2893-7 p. digital

Publication Type: Journal Article

0960-894X

10.1016/s0960-894x(02)00598-x doi


Antineoplastic Agents--chemical synthesis
Cell Line
Cyclization
Enzyme Inhibitors--chemical synthesis
ErbB Receptors--antagonists & inhibitors
Magnetic Resonance Spectroscopy
Mass Spectrometry
Models, Molecular
Molecular Conformation
Nitriles--chemical synthesis
Quinolines--chemical synthesis
Receptor, ErbB-2--antagonists & inhibitors