Sandhu, Sumandeep K

A cocaine insensitive chimeric insect serotonin transporter reveals domains critical for cocaine interaction. [electronic resource] - European journal of biochemistry Aug 2002 - 3934-44 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.

0014-2956

10.1046/j.1432-1033.2002.03084.x doi


Amino Acid Sequence
Animals
Biological Transport--drug effects
Carrier Proteins--antagonists & inhibitors
Cell Line
Chlorides--pharmacology
Chlorocebus aethiops
Cloning, Molecular
Cocaine--pharmacology
Drug Resistance
Fluoxetine--pharmacology
Humans
Hydrophobic and Hydrophilic Interactions
Insect Proteins--antagonists & inhibitors
Manduca--chemistry
Membrane Glycoproteins--antagonists & inhibitors
Membrane Transport Proteins
Molecular Sequence Data
Mutagenesis, Site-Directed
Nerve Tissue Proteins--antagonists & inhibitors
Protein Conformation
Protein Structure, Tertiary
Recombinant Fusion Proteins--antagonists & inhibitors
Sequence Alignment
Sequence Homology, Amino Acid
Serotonin--metabolism
Serotonin Antagonists--metabolism
Serotonin Plasma Membrane Transport Proteins
Serotonin Receptor Agonists--metabolism
Selective Serotonin Reuptake Inhibitors--pharmacology
Sodium--pharmacology
Species Specificity
Structure-Activity Relationship