A cocaine insensitive chimeric insect serotonin transporter reveals domains critical for cocaine interaction. [electronic resource]
- European journal of biochemistry Aug 2002
- 3934-44 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.
0014-2956
10.1046/j.1432-1033.2002.03084.x doi
Amino Acid Sequence Animals Biological Transport--drug effects Carrier Proteins--antagonists & inhibitors Cell Line Chlorides--pharmacology Chlorocebus aethiops Cloning, Molecular Cocaine--pharmacology Drug Resistance Fluoxetine--pharmacology Humans Hydrophobic and Hydrophilic Interactions Insect Proteins--antagonists & inhibitors Manduca--chemistry Membrane Glycoproteins--antagonists & inhibitors Membrane Transport Proteins Molecular Sequence Data Mutagenesis, Site-Directed Nerve Tissue Proteins--antagonists & inhibitors Protein Conformation Protein Structure, Tertiary Recombinant Fusion Proteins--antagonists & inhibitors Sequence Alignment Sequence Homology, Amino Acid Serotonin--metabolism Serotonin Antagonists--metabolism Serotonin Plasma Membrane Transport Proteins Serotonin Receptor Agonists--metabolism Selective Serotonin Reuptake Inhibitors--pharmacology Sodium--pharmacology Species Specificity Structure-Activity Relationship