Levin, Malin C

The myocardium-protective Gly-49 variant of the beta 1-adrenergic receptor exhibits constitutive activity and increased desensitization and down-regulation. [electronic resource] - The Journal of biological chemistry Aug 2002 - 30429-35 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0021-9258

10.1074/jbc.M200681200 doi


Down-Regulation
GTP-Binding Proteins--physiology
Genotype
Glycine
Heart Failure--drug therapy
Humans
Metoprolol--pharmacology
Polymorphism, Genetic
Receptors, Adrenergic, beta-1--chemistry
Structure-Activity Relationship