TY - GEN AU - Gilbert,Adam M AU - Caltabiano,Stephen AU - Koehn,Frank E AU - Chen,Zhen-jia AU - Francisco,Gerardo D AU - Ellingboe,John W AU - Kharode,Yogendra AU - Mangine,AnnaMarie AU - Francis,Rita AU - TrailSmith,Mark AU - Gralnick,David TI - Pyrazolopyrimidine-2,4-dione sulfonamides: novel and selective calcitonin inducers SN - 0022-2623 PY - 2002///0607 KW - 3',5'-Cyclic-AMP Phosphodiesterases KW - antagonists & inhibitors KW - Calcitonin KW - biosynthesis KW - Cell Line KW - Cyclic Nucleotide Phosphodiesterases, Type 4 KW - Genes, Reporter KW - Humans KW - Luciferases KW - genetics KW - Phosphodiesterase Inhibitors KW - chemical synthesis KW - Pyrimidines KW - Radioimmunoassay KW - Structure-Activity Relationship KW - Sulfonamides KW - Transcriptional Activation KW - Xanthines KW - chemistry N1 - Publication Type: Journal Article UR - https://doi.org/10.1021/jm010554s ER -