Gilbert, Adam M

Pyrazolopyrimidine-2,4-dione sulfonamides: novel and selective calcitonin inducers. [electronic resource] - Journal of medicinal chemistry May 2002 - 2342-5 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm010554s doi


3',5'-Cyclic-AMP Phosphodiesterases--antagonists & inhibitors
Calcitonin--biosynthesis
Cell Line
Cyclic Nucleotide Phosphodiesterases, Type 4
Genes, Reporter
Humans
Luciferases--genetics
Phosphodiesterase Inhibitors--chemical synthesis
Pyrimidines--chemical synthesis
Radioimmunoassay
Structure-Activity Relationship
Sulfonamides--chemical synthesis
Transcriptional Activation
Xanthines--chemistry