Martinez, Ana

First non-ATP competitive glycogen synthase kinase 3 beta (GSK-3beta) inhibitors: thiadiazolidinones (TDZD) as potential drugs for the treatment of Alzheimer's disease. [electronic resource] - Journal of medicinal chemistry Mar 2002 - 1292-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-2623

10.1021/jm011020u doi


Adenosine Triphosphate--metabolism
Alzheimer Disease--drug therapy
Amino Acid Sequence
Animals
Binding, Competitive
Calcium-Calmodulin-Dependent Protein Kinases--antagonists & inhibitors
Enzyme Inhibitors--chemical synthesis
Glycogen Synthase Kinase 3
Glycogen Synthase Kinases
Humans
Molecular Sequence Data
Rabbits
Rats
Structure-Activity Relationship
Thiadiazoles--chemical synthesis