Riba, Pal

[Dmt(1)]DALDA is highly selective and potent at mu opioid receptors, but is not cross-tolerant with systemic morphine. [electronic resource] - Current medicinal chemistry Jan 2002 - 31-9 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

0929-8673

10.2174/0929867023371445 doi


Analgesics, Opioid--antagonists & inhibitors
Animals
Drug Tolerance
Enkephalin, Ala(2)-MePhe(4)-Gly(5)---pharmacology
Injections, Intraventricular
Injections, Spinal
Injections, Subcutaneous
Male
Mice
Mice, Inbred ICR
Morphine--administration & dosage
Naloxone--pharmacology
Narcotic Antagonists--pharmacology
Oligopeptides--antagonists & inhibitors
Pain Measurement--drug effects
Receptors, Opioid, mu--agonists
Spinal Cord--drug effects
Time Factors