Identification of novel inhibitors of the transforming growth factor beta1 (TGF-beta1) type 1 receptor (ALK5). [electronic resource]
- Journal of medicinal chemistry Feb 2002
- 999-1001 p. digital
Publication Type: Journal Article
0022-2623
10.1021/jm010493y doi
Activin Receptors, Type I--antagonists & inhibitors DNA-Binding Proteins--metabolism Enzyme Inhibitors--chemical synthesis Fibronectins--biosynthesis Humans Imidazoles--chemical synthesis Mitogen-Activated Protein Kinases--antagonists & inhibitors Protein Serine-Threonine Kinases RNA, Messenger--biosynthesis Receptor, Transforming Growth Factor-beta Type I Receptors, Transforming Growth Factor beta--antagonists & inhibitors Smad3 Protein Structure-Activity Relationship Trans-Activators--metabolism Tumor Cells, Cultured p38 Mitogen-Activated Protein Kinases