Callahan, James F

Identification of novel inhibitors of the transforming growth factor beta1 (TGF-beta1) type 1 receptor (ALK5). [electronic resource] - Journal of medicinal chemistry Feb 2002 - 999-1001 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm010493y doi


Activin Receptors, Type I--antagonists & inhibitors
DNA-Binding Proteins--metabolism
Enzyme Inhibitors--chemical synthesis
Fibronectins--biosynthesis
Humans
Imidazoles--chemical synthesis
Mitogen-Activated Protein Kinases--antagonists & inhibitors
Protein Serine-Threonine Kinases
RNA, Messenger--biosynthesis
Receptor, Transforming Growth Factor-beta Type I
Receptors, Transforming Growth Factor beta--antagonists & inhibitors
Smad3 Protein
Structure-Activity Relationship
Trans-Activators--metabolism
Tumor Cells, Cultured
p38 Mitogen-Activated Protein Kinases