Design, synthesis, and biological activity of methoctramine-related polyamines as putative G(i) protein activators. [electronic resource]
- Journal of medicinal chemistry Nov 2001
- 4035-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-2623
10.1021/jm0155594 doi
Animals Atrial Function CHO Cells Cricetinae Diamines--chemistry Drug Design Electric Stimulation GTP-Binding Protein alpha Subunits, Gi-Go--metabolism Guinea Pigs Heart Atria--drug effects Humans In Vitro Techniques Muscarinic Agonists--pharmacology Polyamines--chemical synthesis Rats Receptors, Muscarinic--metabolism Structure-Activity Relationship