Wang, E

The farnesyl protein transferase inhibitor SCH66336 is a potent inhibitor of MDR1 product P-glycoprotein. [electronic resource] - Cancer research Oct 2001 - 7525-9 p. digital

Publication Type: Journal Article

0008-5472


3T3 Cells--drug effects
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Adenosine Triphosphate--metabolism
Alkyl and Aryl Transferases--antagonists & inhibitors
Animals
Antineoplastic Agents--pharmacology
Biological Transport, Active--drug effects
CHO Cells
Cell Line
Cricetinae
Daunorubicin--pharmacokinetics
Drug Synergism
Enzyme Inhibitors--pharmacology
Farnesyltranstransferase
Genes, MDR
Humans
Hydrolysis
Mice
Paclitaxel--pharmacology
Piperidines--pharmacology
Pyridines--pharmacology
Rhodamine 123--pharmacokinetics
Tamoxifen--pharmacology
Vinblastine--pharmacology