The farnesyl protein transferase inhibitor SCH66336 is a potent inhibitor of MDR1 product P-glycoprotein. [electronic resource]
- Cancer research Oct 2001
- 7525-9 p. digital
Publication Type: Journal Article
0008-5472
3T3 Cells--drug effects ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Adenosine Triphosphate--metabolism Alkyl and Aryl Transferases--antagonists & inhibitors Animals Antineoplastic Agents--pharmacology Biological Transport, Active--drug effects CHO Cells Cell Line Cricetinae Daunorubicin--pharmacokinetics Drug Synergism Enzyme Inhibitors--pharmacology Farnesyltranstransferase Genes, MDR Humans Hydrolysis Mice Paclitaxel--pharmacology Piperidines--pharmacology Pyridines--pharmacology Rhodamine 123--pharmacokinetics Tamoxifen--pharmacology Vinblastine--pharmacology