Statistical molecular design, parallel synthesis, and biological evaluation of a library of thrombin inhibitors. [electronic resource]
- Journal of medicinal chemistry Oct 2001
- 3424-39 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-2623
10.1021/jm010833f doi
Animals Benzenesulfonates--chemical synthesis Binding Sites Cattle Combinatorial Chemistry Techniques Drug Design Humans Magnetic Resonance Spectroscopy Molecular Structure Quantitative Structure-Activity Relationship Serine Proteinase Inhibitors Statistics as Topic Thrombin--antagonists & inhibitors Trypsin--chemistry