Identification of determinants of inverse agonism in a constitutively active parathyroid hormone/parathyroid hormone-related peptide receptor by photoaffinity cross-linking and mutational analysis. [electronic resource]
- The Journal of biological chemistry Nov 2001
- 42692-9 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
0021-9258
10.1074/jbc.M106215200 doi
Animals COS Cells Cattle Cross-Linking Reagents--pharmacology Cyclic AMP--metabolism DNA Mutational Analysis Dose-Response Relationship, Drug Electrophoresis, Polyacrylamide Gel Humans Inhibitory Concentration 50 Leucine--chemistry Ligands Mass Spectrometry Methionine--chemistry Models, Biological Mutagenesis, Site-Directed Mutation Parathyroid Hormone--agonists Peptides--chemistry Plasmids--metabolism Protein Binding Protein Structure, Tertiary Rats Receptors, Parathyroid Hormone--agonists Transfection