Beshore, D C <br/><br/>
Evaluation of amino acid-based linkers in potent macrocyclic inhibitors of farnesyl-protein transferase.  [electronic resource] 

 -  Bioorganic & medicinal chemistry letters  Jul 2001 
 - 1817-21 p.  digital 
<br/><br/> Publication Type: Journal Article 
<br/><br/><label>ISSN: </label>0960-894X 
<br/><br/><label>Standard No.: </label>10.1016/s0960-894x(01)00340-7  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Alkyl and Aryl Transferases--antagonists & inhibitors<br/>Amino Acids--chemistry<br/>Animals<br/>Cells, Cultured<br/>Dogs<br/>Enzyme Inhibitors--administration & dosage<br/>Half-Life<br/>Inhibitory Concentration 50<br/>Metabolic Clearance Rate--physiology<br/>Molecular Conformation<br/>Protein Binding--drug effects<br/>Rats