Bournique, B

In vitro metabolism and drug interaction potential of a new highly potent anti-cytomegalovirus molecule, CMV423 (2-chloro 3-pyridine 3-yl 5,6,7,8-tetrahydroindolizine I-carboxamide). [electronic resource] - British journal of clinical pharmacology Jul 2001 - 53-63 p. digital

Publication Type: Journal Article

0306-5251

10.1046/j.0306-5251.2001.01413.x doi


Adolescent
Adult
Antiviral Agents--metabolism
Biotransformation
Chromatography, High Pressure Liquid
Cytochrome P-450 CYP1A2--metabolism
Cytochrome P-450 CYP1A2 Inhibitors
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--metabolism
Cytomegalovirus--drug effects
Drug Interactions
Enzyme Inhibitors--pharmacology
Female
Humans
Indinavir--metabolism
Indolizines--metabolism
Male
Microsomes, Liver--enzymology
Middle Aged
Mixed Function Oxygenases--antagonists & inhibitors
Molecular Structure
Pyridines--metabolism
Yeasts--enzymology
Zidovudine--metabolism