Giannessi, F

Reversible carnitine palmitoyltransferase inhibitors with broad chemical diversity as potential antidiabetic agents. [electronic resource] - Journal of medicinal chemistry Jul 2001 - 2383-6 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm010889+ doi


3-Hydroxybutyric Acid--blood
Animals
Carnitine--analogs & derivatives
Carnitine O-Palmitoyltransferase--antagonists & inhibitors
Enzyme Inhibitors--chemical synthesis
Hypoglycemic Agents--chemical synthesis
In Vitro Techniques
Mitochondria, Heart--drug effects
Mitochondria, Liver--drug effects
Rats
Rats, Sprague-Dawley
Stereoisomerism
Structure-Activity Relationship