Martin, C

Synthesis of oxa-bridged analogues of farnesyltransferase inhibitor RPR 115135. [electronic resource] - The Journal of organic chemistry Jun 2001 - 3797-805 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-3263

10.1021/jo0100188 doi


Alkyl and Aryl Transferases--antagonists & inhibitors
Bridged-Ring Compounds--chemical synthesis
Cyclization
Enzyme Inhibitors--chemical synthesis
Farnesyltranstransferase
Indicators and Reagents
Indoles
Magnetic Resonance Spectroscopy
X-Ray Diffraction