Contribution of P-glycoprotein to the enhancing effects of dimethyl-beta-cyclodextrin on oral bioavailability of tacrolimus. [electronic resource]
- The Journal of pharmacology and experimental therapeutics May 2001
- 547-55 p. digital
Publication Type: Journal Article
0022-3565
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism Animals Antineoplastic Agents, Phytogenic--pharmacology Area Under Curve Biological Availability Blotting, Western Caco-2 Cells Cyclodextrins--pharmacology Drug Resistance, Neoplasm Flow Cytometry Humans Immunosuppressive Agents--pharmacokinetics Intestinal Absorption--drug effects Male Rats Rats, Wistar Reverse Transcriptase Polymerase Chain Reaction Silver Staining Solubility Tacrolimus--pharmacokinetics Vinblastine--pharmacology beta-Cyclodextrins