TY - GEN AU - Casula,M A AU - Bromidge,F A AU - Pillai,G V AU - Wingrove,P B AU - Martin,K AU - Maubach,K AU - Seabrook,G R AU - Whiting,P J AU - Hadingham,K L TI - Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor SN - 0022-3042 PY - 2001///0517 KW - Amino Acid Sequence KW - Amino Acid Substitution KW - Animals KW - Anti-Anxiety Agents KW - metabolism KW - Azides KW - Benzodiazepines KW - Binding Sites KW - Binding, Competitive KW - Carbolines KW - DNA, Complementary KW - Female KW - Flumazenil KW - Flunitrazepam KW - GABA-A Receptor Agonists KW - Humans KW - Imidazoles KW - Isoleucine KW - chemistry KW - Ligands KW - Molecular Sequence Data KW - Mutagenesis, Site-Directed KW - Oocytes KW - Protein Binding KW - Protein Structure, Tertiary KW - Protein Subunits KW - Pyridazines KW - Pyridines KW - Receptors, GABA-A KW - Recombinant Fusion Proteins KW - Sequence Alignment KW - Structure-Activity Relationship KW - Threonine KW - Transfection KW - Xenopus laevis KW - Zolpidem N1 - Publication Type: Comparative Study; Journal Article UR - https://doi.org/10.1046/j.1471-4159.2001.00289.x ER -