Casula, M A
Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor. [electronic resource]
- Journal of neurochemistry Apr 2001
- 445-51 p. digital
Publication Type: Comparative Study; Journal Article
ISSN: 0022-3042
Standard No.: 10.1046/j.1471-4159.2001.00289.x doi
Subjects--Topical Terms: Amino Acid Sequence Amino Acid Substitution Animals Anti-Anxiety Agents--metabolism Azides--metabolism Benzodiazepines--metabolism Binding Sites Binding, Competitive Carbolines--metabolism DNA, Complementary Female Flumazenil--metabolism Flunitrazepam--metabolism GABA-A Receptor Agonists Humans Imidazoles--metabolism Isoleucine--chemistry Ligands Molecular Sequence Data Mutagenesis, Site-Directed Oocytes Protein Binding Protein Structure, Tertiary Protein Subunits Pyridazines--metabolism Pyridines--metabolism Receptors, GABA-A--chemistry Recombinant Fusion Proteins--chemistry Sequence Alignment Structure-Activity Relationship Threonine--chemistry Transfection Xenopus laevis Zolpidem