TY - GEN AU - Korolkova,Y V AU - Kozlov,S A AU - Lipkin,A V AU - Pluzhnikov,K A AU - Hadley,J K AU - Filippov,A K AU - Brown,D A AU - Angelo,K AU - Strøbaek,D AU - Jespersen,T AU - Olesen,S P AU - Jensen,B S AU - Grishin,E V TI - An ERG channel inhibitor from the scorpion Buthus eupeus SN - 0021-9258 PY - 2001///0510 KW - Amino Acid Sequence KW - Animals KW - Base Sequence KW - Cation Transport Proteins KW - Cell Line KW - Chromatography, High Pressure Liquid KW - Cloning, Molecular KW - DNA, Complementary KW - metabolism KW - DNA-Binding Proteins KW - Dose-Response Relationship, Drug KW - ERG1 Potassium Channel KW - Electrophysiology KW - Escherichia coli KW - Ether-A-Go-Go Potassium Channels KW - Humans KW - Inhibitory Concentration 50 KW - KCNQ Potassium Channels KW - KCNQ1 Potassium Channel KW - Kinetics KW - Mass Spectrometry KW - Mice KW - Molecular Sequence Data KW - Mutagenesis, Site-Directed KW - Mutation KW - Open Reading Frames KW - Polymerase Chain Reaction KW - Potassium Channel Blockers KW - Potassium Channels KW - Potassium Channels, Voltage-Gated KW - Protein Sorting Signals KW - Protein Structure, Tertiary KW - RNA, Messenger KW - Rats KW - Recombinant Fusion Proteins KW - Scorpion Venoms KW - biosynthesis KW - Scorpions KW - Sequence Analysis, DNA KW - Sequence Homology, Amino Acid KW - Substrate Specificity KW - Time Factors KW - Trans-Activators KW - Transcriptional Regulator ERG KW - Tumor Cells, Cultured N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1074/jbc.M005973200 ER -