TY - GEN AU - Dinsmore,C J AU - Zartman,C B AU - Baginsky,W F AU - O'Neill,T J AU - Koblan,K S AU - Chen,I W AU - McLoughlin,D A AU - Olah,T V AU - Huff,J R TI - Synthesis of conformationally constrained 5,6,7, 8-Tetrahydroimidazo[1,5-a]pyridine inhibitors of farnesyltransferase SN - 1523-7060 PY - 2000///1212 KW - Administration, Oral KW - Alkyl and Aryl Transferases KW - antagonists & inhibitors KW - Animals KW - Dogs KW - Enzyme Inhibitors KW - chemical synthesis KW - Farnesyltranstransferase KW - Imidazoles KW - Indicators and Reagents KW - Models, Molecular KW - Molecular Conformation KW - Pyridines KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1021/ol0002424 ER -