White, A W

Resistance-modifying agents. 9. Synthesis and biological properties of benzimidazole inhibitors of the DNA repair enzyme poly(ADP-ribose) polymerase. [electronic resource] - Journal of medicinal chemistry Nov 2000 - 4084-97 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-2623

10.1021/jm000950v doi


Antineoplastic Agents--pharmacology
Benzimidazoles--chemical synthesis
Crystallography, X-Ray
Dacarbazine--analogs & derivatives
Drug Resistance, Neoplasm
Drug Screening Assays, Antitumor
Drug Synergism
Enzyme Inhibitors--chemical synthesis
Humans
Models, Molecular
Poly(ADP-ribose) Polymerase Inhibitors
Structure-Activity Relationship
Temozolomide
Topotecan--pharmacology
Tumor Cells, Cultured