A rational approach to the design and synthesis of a new bradykinin B(1) receptor antagonist. [electronic resource]
- Journal of medicinal chemistry Jun 2000
- 2387-94 p. digital
Publication Type: Journal Article
0022-2623
10.1021/jm990962k doi
Animals Bradykinin Receptor Antagonists CHO Cells Cricetinae Drug Design In Vitro Techniques Magnetic Resonance Spectroscopy Muscle Contraction--drug effects Muscle, Smooth, Vascular--drug effects Oligopeptides--chemical synthesis Receptor, Bradykinin B1 Structure-Activity Relationship Thiazepines--chemical synthesis Transfection Umbilical Veins--drug effects