Expression, characterization and structure determination of an active site mutant (Glu202-Gln) of mini-stromelysin-1. [electronic resource]
- Protein engineering Jun 2000
- 397-405 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
0269-2139
10.1093/protein/13.6.397 doi
Amino Acid Substitution--genetics Aminobiphenyl Compounds--pharmacology Binding Sites--genetics Crystallography, X-Ray Electrophoresis, Polyacrylamide Gel Enzyme Activation--drug effects Enzyme Inhibitors--pharmacology Gelatin--chemistry HeLa Cells Humans Matrix Metalloproteinase 3--biosynthesis Matrix Metalloproteinase Inhibitors Models, Molecular Mutagenesis, Site-Directed Protein Binding--physiology Protein Structure, Tertiary Structure-Activity Relationship Tissue Inhibitor of Metalloproteinase-1--chemistry