TY - GEN AU - Jankun,J AU - Skrzypczak-Jankun,E TI - Molecular basis of specific inhibition of urokinase plasminogen activator by amiloride SN - 0305-7232 PY - 2000///0802 KW - Amiloride KW - chemistry KW - Amino Acid Chloromethyl Ketones KW - Amino Acid Sequence KW - Antineoplastic Agents KW - Binding Sites KW - drug effects KW - Binding, Competitive KW - Catalysis KW - Crystallography, X-Ray KW - Drug Design KW - Humans KW - Models, Molecular KW - Molecular Conformation KW - Molecular Sequence Data KW - Neoplasm Proteins KW - antagonists & inhibitors KW - Protein Binding KW - Protein Conformation KW - Protein Structure, Tertiary KW - Sequence Alignment KW - Sequence Homology, Amino Acid KW - Serine Proteinase Inhibitors KW - Substrate Specificity KW - Tissue Plasminogen Activator KW - Urokinase-Type Plasminogen Activator KW - Water N1 - Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't ER -