Jankun, J

Molecular basis of specific inhibition of urokinase plasminogen activator by amiloride. [electronic resource] - Cancer biochemistry biophysics Jul 1999 - 109-23 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

0305-7232


Amiloride--chemistry
Amino Acid Chloromethyl Ketones--chemistry
Amino Acid Sequence
Antineoplastic Agents--chemistry
Binding Sites--drug effects
Binding, Competitive
Catalysis--drug effects
Crystallography, X-Ray
Drug Design
Humans
Models, Molecular
Molecular Conformation
Molecular Sequence Data
Neoplasm Proteins--antagonists & inhibitors
Protein Binding
Protein Conformation
Protein Structure, Tertiary
Sequence Alignment
Sequence Homology, Amino Acid
Serine Proteinase Inhibitors--chemistry
Substrate Specificity
Tissue Plasminogen Activator--chemistry
Urokinase-Type Plasminogen Activator--antagonists & inhibitors
Water--chemistry