Schiller, P W

Novel ligands lacking a positive charge for the delta- and mu-opioid receptors. [electronic resource] - Journal of medicinal chemistry Feb 2000 - 551-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0022-2623

10.1021/jm990461z doi


Animals
Binding, Competitive
Brain--metabolism
Guinea Pigs
Ileum--drug effects
In Vitro Techniques
Ligands
Male
Mice
Muscle Contraction--drug effects
Muscle, Smooth--drug effects
Narcotic Antagonists--chemical synthesis
Neurokinin-1 Receptor Antagonists
Oligopeptides--chemical synthesis
Peptides, Cyclic--chemical synthesis
Radioligand Assay
Rats
Receptors, Neurokinin-1--metabolism
Receptors, Opioid, mu--antagonists & inhibitors
Structure-Activity Relationship
Vas Deferens--drug effects