Perloff, M D

Midazolam and triazolam biotransformation in mouse and human liver microsomes: relative contribution of CYP3A and CYP2C isoforms. [electronic resource] - The Journal of pharmacology and experimental therapeutics Feb 2000 - 618-28 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

0022-3565


Animals
Antibodies--pharmacology
Aryl Hydrocarbon Hydroxylases
Biotransformation
Blotting, Western
Chromatography, High Pressure Liquid
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme System--immunology
Dose-Response Relationship, Drug
Humans
Immunochemistry
In Vitro Techniques
Inhibitory Concentration 50
Ketoconazole--pharmacology
Mice
Microsomes, Liver--metabolism
Midazolam--pharmacokinetics
Mixed Function Oxygenases--immunology
Oxidoreductases, N-Demethylating--physiology
Protein Isoforms--physiology
Species Specificity
Steroid 16-alpha-Hydroxylase
Steroid Hydroxylases--immunology
Triazolam--pharmacokinetics